2020
Tarek S Ibrahim, Mohamed M Hawwas, Ehab S Taher, Nabil A Alhakamy, Mohamed A Alfaleh, Mohamed Elagawany,
Bahaa Elgendy, Gamal M Zayed, Mamdouh FA Mohamed, Zakaria K Abdel-Samii, Yaseen AMM Elshaier.
Design and synthesis of novel pyrazolo [3, 4-d] pyrimidin-4-one bearing quinoline scaffold as potent dual PDE5 inhibitors and apoptotic inducers for cancer therapy.
Bioorg. Chem., 2020,105, 104352
Mohamed Shahien, Mohamed Elagawany, Sadichha Sitaula, Shaimaa S Goher, Sheryl L Burris, Ryan Sanders, Amer Avdagic, Cyrielle Billon, Lamees Hegazy, Thomas P Burris,
Bahaa Elgendy*.
Modulation of estrogen-related receptors subtype selectivity: Conversion of an ERRβ/γ selective agonist to ERRα/β/γ pan agonists. Bioorg. Chem., 2020,102, 104079.
Elzahhar, P. A.; Abd El Wahab, S. M.; Elagawany, M.; Daabees, H.; Belal, A.; EL-Yazbi, A.; Eid, A.; Alaaeddine, R.; Hegazy, R.; Allam, R.; Helmy, M.;
Elgendy, B.; Angeli, A.; El-Hawash, S.; Supuran, C. T.
Expanding the anticancer potential of 1,2,3-triazoles via simultaneously targeting Cyclooxygenase-2, 15-lipoxygenase and tumor-associated carbonic anhydrases. Eur. J. Med. Chem. 2020, 200, 112439.
Ibrahim, T. S.; Salem, I. M.; Mostafa, S. M.; El-Sabbagh, O. I.; ElKhamisi, M. K.; Hegazy, L.;
Elgendy, B*. Design, synthesis, and pharmacological evaluation of novel and selective COX-2 inhibitors based on bumetanide scaffold. Bioorg. Chem., 2020, 100, 103878.
Saeed, W.; Elagawany, M.; Azab, M. M.; Amin, A. S.; Rath, N. P.; Hegazy, L.;
Elgendy, B*. Catalyst-and organic solvent-free synthesis, structural, and theoretical studies of 1-arylidenamino-2,4-disubstituted-2-imidazoline-5-ones. Results in Chemistry 2020, 2, 100042.
2019
Goher, S.S.; Griffett, K.; Hegazy, L.; Elagawany, M.; Arief, M.M.H.; Avdagic, A.; Banerjee, S.; Burris, T.P.;
Elgendy, B*. Development of novel liver X receptor modulators based on a 1,2,4-triazole scaffold. Bioorg. Med. Chem. Lett., 2019, 29 (3), 449-453.
2018
Cao, F.; Orth, C.; Donlin, M.J.; Adegboyega, P.; Meyers, M.J.; Murelli, R.P.; Elagawany, M.;
Elgendy, B.; Tavis, J.
Synthesis and evaluation of troponoids as a new class of antibiotics. ACS Omega, 2018, 3 (11), 15125-15133.
Elagawany, M.; Hegazy, L.; Cao, F.; Donlin, M.J.; Rath, N.; Tavis, J.;
Elgendy, B*.
Identification of 4-isopropyl–thiotropolone as a novel anti-microbial: regioselective synthesis, NMR characterization, and biological evaluation. RSC Advances, 2018, 8 (52), 29967-29975.
El-Sayed, S.; Ali, M.;
Elgendy, B.; Dandash, S.; Issac, Y.; Saad, R.; Azab, M.; Mohamed, M.
Identification of novel small molecule inhibitors against the NS3/4A protease of hepatitis C virus genotype 4a.
Curr. Pharm. Des., 2018, 24 (37), 4484-4491.
2016
Mabied, A.F.; Girgis, A.S.; Shalaby, E.M.; George, R.F.;
Elgendy, B.; Baseliouse, F.N.
Stereoselective Synthesis, Structural and Spectroscopic Study of 4,5,11-Triazatricyclo[6.2.1.0*2,6*]Undec-5-ene. J. Heterocyclic Chem., 2016, 53, 1074-1080.
2015
Flaveny, C.A.; Griffett, K.;
Elgendy, B.; Kazantzis, M. Sengupta, M.; Amelio, A.L.; Chatterjee, A.; Walker, J.; Solt, L.A.; Kamenecka, T.M.; Burris, T.P.
Broad Anti-Tumor Activity of a Small Molecule that Selectively Targets the Warburg Effect and Lipogenesis. Cancer Cell, 2015, 28 (1), 42-56.
2014
Shalaby, E.M.; Girgis, A.S.; Moustafa, A.M.; ElShaabiny, A.M.;
Elgendy, B.; Mabied, A.F.; Farag, I.S. A.
Regioselective Synthesis, Stereochemical Structure, Spectroscopic Characterization and Geometry Optimization of Dispiro[3H-Indole-3,2′-Pyrrolidine-3′,3′′-Piperidines].
J. Mol. Struct., 2014, 1075, 327–334.
2013
Khan, P.M.;
Elgendy, B.; Kumar, N.; Chang, M.R.; Lin, L.; Ruiz, C.H.; Cameron, M.D.; Griffin, P.R.; Kamenecka, T.M.
Small Molecule Amides as Potent ROR-γ Selective Modulators.
Bioorg. Med. Chem. Lett., 2013, 23, 532-536.
2012
Draghici, B.;
Elgendy, B.; Katritzky, A.R.
Synthesis of Benzoxazines, Quinazolines and 4H-Benzo[e][1,3]thiazine by ANRORC Rearrangements of 1,2,4-Oxadiazoles.
Synthesis, 2012, 44, 547–550.
Ghazvini Zadeh, E.H.;
Elgendy, B.; Pop, A.G.; Katritzky, A.R.
Synthesis of chiral α-amino acid-derived 1H-1,2,4-triazoles and 1,2,4-triazines.
Med. Chem. Commun., 2012, 3, 52-55.
2011
Hall, A.C.; Griffith, T.N.; Tsikolia, M..; Kotey, F.O.; Gill, N.; Humbert, D.J.; Watt, E.E.; Yermolina, Y.A.; Goel, S.;
Elgendy, B.; Hall, C.D.
Cyclohexanol Analogues are Positive Modulators of GABAA Receptor Currents and Act as General Anaesthetics in Vivo.
Eur. J. Pharmacol. 2011, 667, 175–181.
2010
Katritzky, A.R.;
Elgendy, B.; Draghici, B.; Fedoseyenko, D.; Fadli, A.; Metais, E.
1H, 13C, and 15N NMR Spectra of Some Pyridazine Derivatives. Magn. Reson. Chem. 2010, 48(5), 397-402.
2009
2008
2007